Formal Total Synthesis of Manzacidin B via Sequential Diastereodivergent Henry Reaction
نویسندگان
چکیده
منابع مشابه
Total synthesis of calothrixin B via sequential Sonogashira coupling/copper-catalyzed oxidative cyclization.
A total synthesis of the antimalarial indolo[3,2-j]phenanthridine alkaloid calothrixin B is reported. The key intermediate, ketoester 11, was assembled using sequential Sonogashira coupling and intra/intermolecular fashioned copper-catalyzed oxidative cyclization reactions.
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ژورنال
عنوان ژورنال: The Journal of Organic Chemistry
سال: 2019
ISSN: 0022-3263,1520-6904
DOI: 10.1021/acs.joc.9b02811